Active Pharmaceutical Ingredient

Rilmenidine — CAS 87333-19-5

Also known as: Tenaxum; S3341; Hyperium

GMP Certified IP / BP / EP / USP Antihypertensive / Imidazoline Receptor Agonist Aurangabad, India
Rilmenidine API Supplier Manufacturer Aurangabad Maharashtra India — Mediocon Inc
Rilmenidine IP / BP / EP / USP  |  GMP Certified  |  Mediocon Inc, Maharashtra, India
CAS No: 87333-19-5

Product Overview

Rilmenidine is a high-purity Active Pharmaceutical Ingredient (API) classified as an Antihypertensive and Imidazoline receptor agonist. Mediocon Inc manufactures GMP-compliant Rilmenidine at its facility in Aurangabad, Maharashtra, India.

Therapeutic Applications
  • Management of essential hypertension
  • Central sympatholytic blood pressure reduction
  • Imidazoline I1 receptor research
  • Combination antihypertensive regimens

Technical Specifications

ParameterSpecification
CAS Number87333-19-5
Molecular FormulaC₉H₁₅N₃O
Molecular Weight181.24 g/mol
GradeIP / BP / EP / USP
CategoryAntihypertensive / Imidazoline Receptor Agonist
AssayNLT 98.0%
Loss on DryingNMT 0.5%
Heavy MetalsNMT 20 ppm
Residue on IgnitionNMT 0.1%
Microbial LimitsComplies with pharmacopoeia
IdentificationIR, HPLC Compliant
Batch NoRLM/24032026
Mfg DateMAR 2026
Exp DateFEB 2031
Packing25 kg HDPE drums / as per requirement

Quality & Compliance

  • GMP Certified manufacturing facility in Aurangabad, Maharashtra, India
  • Full pharmacopoeial compliance: IP / BP / EP / USP standards
  • Complete documentation: Certificate of Analysis (CoA), MSDS, Certificate of Origin
  • Stringent in-process quality control at every manufacturing stage
  • HPLC purity testing and spectroscopic identification (IR, NMR)
  • Cold-chain and controlled-environment storage facilities available
  • Exported to 40+ countries with full regulatory support
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