Active Pharmaceutical Ingredient

Linagliptin

Also known as: Tradjenta; BI 1356

CAS: 668270-12-0 DPP-4 Inhibitor / Antidiabetic IP / BP / EP / USP GMP Certified Aurangabad, Maharashtra, India
Linagliptin API — Mediocon Inc
Linagliptin — Pharmaceutical Grade API

Product Overview

CAS No: 668270-12-0  |  MF: C₂₅H₂₈N₈O₂  |  MW: 472.54 g/mol

Linagliptin is a pharmaceutical-grade active ingredient classified as DPP-4 Inhibitor / Antidiabetic. Mediocon Inc supplies high-purity Linagliptin API conforming to IP / BP / EP / USP specifications, manufactured in our GMP-certified facility in Aurangabad, Maharashtra, India.

Key Features

  • DPP-4 inhibitor antidiabetic
  • IP/BP/EP/USP compliant
  • Full CoA and MSDS documentation
  • GMP certified manufacturing

Applications

  • Type 2 diabetes mellitus management
  • Combination antidiabetic therapy
  • Cardiovascular risk reduction in diabetics

Why Choose Mediocon

  • ISO 9001:2015 & GMP certified manufacturing
  • Consistent batch-to-batch quality with full CoA
  • Export-ready documentation: COO, MSDS, DMF
  • Flexible MOQ for both R&D and commercial scale
  • Dedicated QA support for regulatory filings

Product Specifications

Product NameLinagliptin
Also Known AsTradjenta; BI 1356
CAS Number668270-12-0
Chemical NameLinagliptin
Molecular FormulaC₂₅H₂₈N₈O₂
Molecular Weight472.54 g/mol
CategoryDPP-4 Inhibitor / Antidiabetic
AppearanceWhite to yellowish white crystalline powder
SolubilitySlightly soluble in water, soluble in dimethylformamide
GradeIP / BP / EP / USP

Analytical Specifications

ParameterSpecification
AssayNLT 98.0%
Loss on DryingNMT 0.5%
Heavy MetalsNMT 20 ppm
Residue on IgnitionNMT 0.1%
Microbial LimitsComplies with pharmacopoeia
IdentificationIR, HPLC Compliant
Packing25 kg HDPE drums / as per requirement
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